D3/5-HT receptor modulator-1 [898532-85-9]
Cat# T205297-5mg
Size : 5mg
Marca : TargetMol
D3/5-HT receptor modulator-1
Copy Product InfoD3/5-HT receptor modulator-1 (compound 5i) is a selective antagonist of the dopamine D3 and 5-HT2A receptors, and a partial agonist at the 5-HT1A receptor. It exhibits Ki values of 4.5 nM, 11.9 nM, and 15.3 nM for the dopamine D3, 5-HT2A, and 5-HT1A receptors respectively. The compound shows lower affinity for the dopamine D2 receptor, 5-HT2C receptor, and hERG channel. D3/5-HT receptor modulator-1 possesses atypical antipsychotic properties.
Cas No. 898532-85-9
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Product Information
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | D3/5-HT receptor modulator-1 (compound 5i) is a selective antagonist of the dopamine D3 and 5-HT2A receptors, and a partial agonist at the 5-HT1A receptor. It exhibits Ki values of 4.5 nM, 11.9 nM, and 15.3 nM for the dopamine D3, 5-HT2A, and 5-HT1A receptors respectively. The compound shows lower affinity for the dopamine D2 receptor, 5-HT2C receptor, and hERG channel. D3/5-HT receptor modulator-1 possesses atypical antipsychotic properties. |
| Targets & IC50 | ERG channel (human):930 nM(Ki) |
| Molecular Weight | 391.506 |
| Formula | C24H29N3O2 |
| Cas No. | 898532-85-9 |
| Smiles | O=C(NCCCCN1CCN(C2=CC=CC(=C2)C)CC1)C=3OC=4C=CC=CC4C3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |